I-Raw Orlistat powder (ividiyo ye-96829-58-2)
I-Orlistat powder emnyama (96829-58-2)
I-Raw Orlistat powder isekilasini lemithi ebizwa nge-lipase inhibitors esebenza ngokuvimba ukumuncwa kwamafutha angama-25% esidlweni futhi isetshenziselwa ukwehlisa isisindo kubantu abadala abakhuluphele ngokweqile, abaneminyaka engu-18 nangaphezulu, uma isetshenziswa kanye ne-kilojoule encishisiwe ukudla okunamafutha amancane. I-Raw Orlistat powder isidakamizwa esenzelwe ukwelapha ukukhuluphala. Umsebenzi wawo oyinhloko ukuvimbela ukumuncwa kwamafutha kusuka ekudleni komuntu, ngaleyo ndlela kunciphise ukungena kwe-caloric. I-Raw Orlistat powder isebenza ngokuvimbela i-pancreatic lipase, i-enzyme ephula i-triglycerides emathunjini. Ngaphandle kwale enzyme, ama-triglycerides asuka ekudleni avinjelwe ekungenisweni yi-hydrolyzed ibe ngama-fatty acids angenakutholwa futhi akhishwe angadliwe. I-Prescription Raw Orlistat powder isetshenziswa kubantu abakhuluphele kakhulu abangase babe nengcindezi ephezulu yegazi, isifo sikashukela, i-cholesterol ephezulu, noma isifo senhliziyo. Ukusebenza kwe-Raw Orlistat powder ekukhuthazeni ukulahleka kwesisindo kucacile kepha kunesizotha. Idatha ehlanganisiwe evela ekuhlolweni kwemitholampilo iphakamisa ukuthi abantu banikezwe i-Raw Orlistat powder ngaphezu kokuguqulwa kwendlela yokuphila, njengokudla nokuzivocavoca umzimba, balahlekelwa cishe ngama-2-3 kilograms (4.4-6.6 lb) ngaphezu kwalabo abangathathi umuthi phakathi nonyaka. I-Raw Orlistat powder nayo ngesizotha inciphisa umfutho wegazi futhi ibonakale ivimbela ukuqala kohlobo lwesifo sikashukela sohlobo lwe-2, kungaba kusuka ekulahlekelweni kwesisindo uqobo noma eminye imiphumela. Kunciphisa izehlakalo zesifo sikashukela sohlobo II kubantu abakhuluphele ngokulingana nenani elifanayo noshintsho lwendlela yokuphila.
I-Orlistat powder emnyama (Imininingwane ye-96829-58-2)
Igama Product | I-Orlistat powder |
Igama leKhemikhali | Tetrahydrolipstatin, 1-((3-hexyl-4-oxo-2-oxetanyl)methyl)dodecyl-2-formamido-4-methylvalerate |
Brand NAme | I-Alli, i-Xenical |
I-Drug Class | lipase inhibitors |
CAS Inombolo | 96829-58-2 |
InChIKey | AHLBNYSZXLDEJQ-FWEHEUNISA-N |
I-molecular Fi-ormula | C29H53NO5 |
I-molecular Weziyisishiyagalombili | I-495.745 g / mol |
IMisa ye-Monoisotopic | I-495.392 g / mol |
Ukuxuba Pi-oint | <50 ° C |
Fukuvuselela kabusha Pi-oint | Ayikho idethi etholakalayo |
I-Half Half-Life | Ngokusekelwe kwedatha elinganiselwe, ingxenye yokuphila ye-Raw Orlistat powder etholakalayo iphakathi kwe-1 namahora we-2. |
Color | powder emhlophe |
solubility | I-DMSO: 19 mg / mL |
Storage Tukushisa | Isikhathi sokugcina. I-2-8 ° C |
Aukuphikisana | Sebenzisa ukuphatha ukukhuluphala. |
I-Orlistat emifushane i-powder (96829-58-2) Incazelo
I-Orlistat powder ewomshini elasini lemithi ebizwa ngokuthi i-lipase inhibitors esebenza ngokuvimbela ukumunwa kwe-25% wamafutha esidlweni futhi isetshenziselwa ukulahlekelwa isisindo kubantu abadala abakhuluphele, iminyaka engu-18 nangaphezulu, uma isetshenziselwa ne-calori encishisiwe futhi ukudla okunamafutha aphansi.
I-Orlistat powder ewomshini yidakamizwa eyenzelwe ukwelapha ukukhuluphala. Umsebenzi wayo oyinhloko uvimbela ukungenisa amafutha ekudleni komuntu, ngaleyo ndlela kuncishiswe ukudla kwe-caloric. I-Orlistat powder ewomshini isebenza ngokuvimbela i-pancreatic lipase, i-enzyme ephula i-triglycerides emathunjini. Ngaphandle kwalokhu ku-enzyme, i-triglycerides kusukela ekudleni ivinjelwe ekubeni i-hydrolyzed ibe yi-fatty acids free acids futhi ixhunyiwe ngaphandle kwe-nongested. I-Orlistat powder ye-prescription eqoshiwe isetshenziselwa abantu abaqine ngokweqile abangase babe nomfutho wegazi ophezulu, isifo sikashukela, i-cholesterol ephakeme noma isifo senhliziyo. Ukuphumelela kwe-Raw Orlistat powder ekukhuthazeni ukulahlekelwa kwesisindo kuqondile kepha kuthobekile. Idatha ehlukanisiwe kusuka ekuhlolweni kwemitholampilo iphakamisa ukuthi abantu banikezwa i-Orwolat e-Radiat ephuzile ngaphezu kokuguqula indlela yokuphila, njengokudla nokuzivocavoca, balahlekelwa ngamakhilogremu angu-2-3 (4.4-6.6 lb) ngaphezu kwalabo abangathathi izidakamizwa phakathi nenkathi yonyaka. I-Orlistat powder enqamulelayo futhi iyancipha ngokunciphisa ukucindezeleka kwegazi futhi ibonakala ivimbela ukuqala kohlobo lwe-2 yesifo sikashukela, kungakhathaliseki ukuthi isisindo sokulahlekelwa ngokwayo noma eminye imiphumela. Linciphisa izifo zesifo sikashukela uhlobo II kubantu abakhuluphele abazungeze inani elifanayo lokuthi izinguquko zokuphila zenzani.
I-Orlistat powder (96829-58-2) Indlela Yokusebenza
I-Orlistat powder uhlobo lwe-lipase oluvimbela izidakamizwa zokulahlekelwa isisindo futhi luyisithako esivela ku-lipostatin. I-Orlistat ivimbela ngempumelelo futhi ngokukhetha isisu se-lipase ne-pancreatic lipase, ngenkathi ingenawo umthelela kwamanye ama-enzyme wokugaya ukudla (njenge-amylase, i-trypsin ne-chymotrypsin) kanye ne-phospholipase, futhi ayikuthinti ukumuncwa kwama-carbohydrate, amaprotheni kanye ne-phospholipids. Lesi sidakamizwa asimunciwe noma ngabe umgudu wamathumbu futhi sinomphumela wokuvimbela oguqukayo ku-lipase. I-Orlistat ivimbela ama-enzyme ngokubopha okuhlanganayo kokusalele kwe-serine ezindaweni ezisebenzayo zesisu ne-pancreatic lipase. Lokhu kuvimbela amafutha ekudleni ukuthi angahlukaniswa abe ngama-acid anamahhala kanye ne-diacylglycerol, ngakho-ke ayikwazi ukumuncwa, yehlise ukudla kwe-caloric ngakho-ke ilawule isisindo somzimba. Lesi sidakamizwa asidingi ukuthi simunceke umzimba wonke ukuze sisebenze. Umsebenzi we-Orlistat wemithi uncike kumthamo: isilinganiso sokwelashwa se-Orlistat (i-120mg / d, i-tid, ethathwe nokudla), kuhlanganiswe nokudla okunama-khalori aphansi, kunganciphisa ukufika ku-30% wokumunca amafutha. Esifundweni esiqhathanisa amavolontiya ajwayelekile futhi akhuluphele ngokweqile, i-Orlistat empeleni yayingamuncwanga umzimba nhlobo futhi yayinokuhlushwa kwegazi okuphansi kakhulu. Ngemuva kwesilinganiso esisodwa somlomo (esikhulu kunazo zonke singu-800mg), ukuhlanganiswa kwegazi kwe-Orlistat kulawa mahora alandelayo ayi-8 kwakungu- <5 ng / ml. Imvamisa, isilinganiso sokwelashwa se-Orlistat simuncwa umzimba kuphela futhi ngeke siqongeleleke ngesikhathi esifushane sokwelapha. Ekuhlolweni kwe-in vitro, isilinganiso sokubopha se-Orlistat namanye amaprotheni we-serum seqe ama-99% (amaprotheni aboshiwe ikakhulukazi ama-lipoprotein ne-albhamuin), futhi isilinganiso salo sokubopha ngamaseli abomvu egazi sasiphansi kakhulu.
Izinzuzo ze-Orlistat powder (96829-58-2)
Or I-Orlistat inciphisa isisindo somzimba ngamaphesenti angaphezu kuka-20 ngemali yamafutha omzimba
▪ I-Orlista ikusiza ukuthi ufunde ukubala ama-calories
▪ I-Orlista ikunikeza umuzwa wenhlalakahle
▪ I-Orlista inemiphumela emihle enikeza ukuzethemba nenjabulo kubasebenzisi
▪ I-Orlista inikeza imiphumela yesikhathi eside esimeme
▪ I-Orlista inciphisa ubucayi bezifo ezifana ne-hypotension, isifo sikashukela, i-atherosclerosis kanye
i-cholesterol.
I-Orlistat enconyiwe i-powder (96829-58-2) Isilinganiso
Umthamo ophakanyisiwe we-Orlistat powder ungenye ye-120-mg capsule kathathu ngosuku ngokudla okuyinhloko okuqukethe amafutha (ngesikhathi noma kuze kufike ku-1 ihora ngemva kokudla). Amanani angaphezulu kwe-120 mg kathathu ngosuku awabonwanga ukunikeza inzuzo eyengeziwe.
Abantu kufanele babe nokudla okunomsoco, okunciphise-ikhalori okuqukethe cishe ama-30% wamakorikhi avela kumafutha. Ukudla kwansuku zonke kwamafutha, ama-carbohydrate, kanye namaprotheni kufanele kusakazwe ngaphezu kwezidlo ezintathu eziyinhloko. Uma ukudla kungabanjwanga ngezinye izikhathi noma kungaqukethe amafutha, umthamo we-Orlistat powder ungashiywa.
Ngenxa yokuthi i-Orlistat powder ikhonjisiwe ukunciphisa ukumuncwa kwamavithamini ancibilika ngamafutha kanye ne-betacarotene, abantu kufanele belulekwe ngokuthi bathathe i-multivitamin equkethe amavithamini ancibilika amafutha ukuqinisekisa ukudla okwanele. Ngaphandle, isithasiselo sevithamini kufanele sithathwe okungenani amahora we-2 ngaphambi noma ngemuva kokuphathwa kwe-Orlistat powder, njengesikhathi sokulala.
Imiphumela emibi ye-Orlistat powder (96829-58-2)
Kuyinto evamile ukubona imiphumela emibi ye-Orlistat powder uma usisebenzisa. Ungase ubone ezinye imiphumela emibi noma hhayi nje emva kokuthatha noma yimiphi imithi. Iningi lemiphumela efika nokusetshenziswa kwe-Orlistat powder kuhlobene nendlela isebenza ngayo ohlelweni lwakho lokugaya. Ngokuvamile ziba mnene futhi zenzeke njalo uma uqala ukwelashwa. Kwenzeka futhi ngemuva kokuba uthathe ukudla okunamafutha aphezulu. Ngenhlanhla, iningi labo lihamba njengoba ukwelashwa kuqhubeka futhi ngemva kokulandela ukudla okulungile.
Okulandelayo yiminye imiphumela emibi ejwayelekile:
▲ bekhanda
▲ Ubuhlungu besisu / ukuphazamiseka
▲ Ukukhishwa kwamafutha
▲ Izitshalo ezinamafutha
▲ Ukushisa isikhumba esincane
▲ Ukuhlungu obusemhlane
Ngaphandle kwalokho, uma uthola noma yimuphi wale mibi, kufanele uyiphathe njengesimo esiphuthumayo bese ushayele udokotela ngokushesha. Kunjalo;
▲ Ubuhlungu obukhulu besisu obungaphumi.
▲ I-hives noma ukushaya ngokweqile
▲ Kunzima ukugwinya
▲ Ukuphefumula okunzima