I-Raw Tianeptine powder (66981-73-5)

I-Raw Tianeptine powder (66981-73-5) ividiyo

I-Raw Tianeptine powder (66981-73-5)

I-Raw Tianeptine powder iyinhlangano ephikisana nokucindezeleka enephrofayli ye-neurochemical novel. I-Raaw Tianeptine powder ayibonakali ihlotshaniswa nokuhlukumezeka kwengqondo, ingqondo, ukulala, imiphumela ye-cardiovascular noma ye-bodyweight futhi inomzimba ophansi wokuhlukunyezwa. I-Raw Tianeptine powder inephrofayli ye-pharmacokinetic ehle kakhulu. Akuhambisani nokuqala kwesimiso se-hepatic, esine-bioavailability ephezulu nokusabalalisa okulinganiselwe, futhi isuswa ngokushesha. Nakuba lokhu kunikeza izinzuzo ze-Raw Tianeptine powder phezu kwama-tricyclic anti-depressant agents ngokusho kwe-dose, izinguquko zokwelashwa kanye nokusebenzisana kwezidakamizwa okungenzeka, ukususwa kwayo ngokushesha kwenza ukunamathela kwamashejuli amaminithi kubaluleke nakakhulu. I-Raw Tianeptine i-powder ihluke kuningi lezinkinga zokulwa nokucindezeleka ngoba akuyona imetabolised uhlelo olusha lwe-cytochrome P450, olubonisa amathuba amancane okusebenzisana kwezidakamizwa; lokhu kunesithakazelo ngokukhethekile iziguli ezigugile.

I-Raw Tianeptine powder (66981-73-5) Imininingwane

I-Raw Tianeptine powder (66981-73-5) Incazelo

I-Tianeptine powder iyisidakamizwa esetshenziswa kakhulu ekuthuthukiseni izimpawu zengcindezi enkulu yokucindezeleka (MDD). Kuye kwasetshenziselwa ukusiza ukucasula isifo sofuba nesifo se-asthma. Ngokwemvelo, ihlukaniswa ngokuthi i-tricyclic antidepressant (TCA), noma kunjalo, inempahla ehlukile yezokwelapha kunezindlela ezivamile zokulwa nokucindezeleka kwama-tricyclic. I-Tianeptine yatholakale futhi yenziwe i-patented ngumphakathi waseFrance wezokwelapha kwezokwelapha ku-1960s. Amagama omkhiqizo afaka iStablon, Coaxil. ITatinol, Tianeurax, neSalymbra.

I-tianeptine powder ayibonakali ihlotshaniswa nokuhlukumezeka okungaqondakali, ingqondo, ukulala, imiphumela ye-cardiovascular noma bodyweight futhi inomthamo ophansi wokuhlukunyezwa. I-Raw Tianeptine powder inephrofayli ye-pharmacokinetic ehle kakhulu. Akuhambisani nokuqala kwesimiso se-hepatic, esine-bioavailability ephezulu nokusabalalisa okulinganiselwe, futhi isuswa ngokushesha. Nakuba lokhu kunikeza izinzuzo ze-Raw Tianeptine powder phezu kwama-tricyclic anti-depressant agents ngokusho kwe-dose, ukuguqulwa kokwelashwa kanye nokusebenzisana kwezidakamizwa okungenzeka, ukususwa kwayo ngokushesha kwenza ukunamathela kumashejuli amaminithi kubaluleke nakakhulu. I-Raw Tianeptine i-powder ihluke kuningi lezinkinga zokulwa nokucindezeleka ngoba akuyona imetabolised uhlelo olusha lwe-cytochrome P450, olubonisa amathuba amancane okusebenzisana kwezidakamizwa; lokhu kunesithakazelo ngokukhethekile iziguli ezigugile.

Muva nje, i-Tianeptine iyatholakala emazweni aseYurophu, ase-Asia, naseNingizimu Melika. Ivinjelwe e-United Kingdom futhi ayinakekelwa ngokomuthi odokotela base-United States.

I-Tianeptine powder (66981-73-5) Indlela Yokusebenza

Ucwaningo lwamuva lubonisa ukuthi i-tianeptine isebenza njenge-agonist egcwele ku-receptionor ye-opioid (MU). I-receptors yama-opioid njengamanje ihlolisiswa njengenhloso ephumelelayo yezokwelapha ezicindezelayo. Kukholelwa ukuthi imiphumela yomtholampilo ye-tianeptine inesidingo sokuguquguquka kwayo kwala ma-receptors. Ngaphezu kwezinyathelo zawo kwi-receptor ye-opioid, izifundo zangaphambilini zikhokhelwe isenzo salo kumphumela we-serotonin receptor dopamine (D2 / 3) nama-receptors we-glutamate.

I-Tianeptine powder iyimithi ekhethekile yokucindezeleka nokucindezeleka eyenza ukutholakala kwe-serotonin (i-5-hydroxytryptamine; i-5-HT), ne-5-hydroxyindoleacetic acid (i-5-HIAA) emathisini ebuchopho.

Nakuba i-serotonin ye-monoaminergic neurotransmitters (i-5-HT), i-noradrenaline (NA) ne-dopamine (DA) ikhonjiswe ukuthi ihlobene nokuvela kwezinkinga zokucindezeleka, manje sekuqaphele ukuthi ukulahlekelwa kwe-monoamine akwanele ukuchaza indlela yokwenza i-anti-depressant imithi.

Isicelo se-Tianeptine powder (i-66981-73-5)

▪ I-Tianeptine ithuthukisa izimpawu zokucindezeleka okukhulu (MDD)

▪ Usizo lwe-Tianeptine olukhubaza isifo sofuba nesifo se-asthma

▪ I-Tianeptine ithuthukisa isimo sengqondo futhi ikhuthaza ukukhathazeka.

▪ I-Tianeptine yandisa ukuthi isifo se-serotonin sithatha kangakanani

▪ I-Tianeptine ithuthukisa ukugqugquzela, ukugxila nokuqonda, ukunqanda ukukhathazeka, ukuvuselelwa nokunciphisa ukukhathala okungqondweni.

Kunconywe i-Tianeptine powder (i-66981-73-5) Isilinganiso

I-tianeptine powder ngokuvamile ibhalwe ngomthamo we-12.5 mg futhi ithathwa kathathu ngosuku. Ngokungafani namanye ama-TCA kanye nama-serotonin reuptake inhibitors (SSRIs) akhethiwe, ama-tianeptine amanani akudingeki akhuliswe kancane futhi i-taper uma imithi ishiyiwe ayidingekile.

Imiphumela emibi ye-Tianeptine powder (66981-73-5)

Imiphumela emibi ye-tianeptine powder iyamangalisa kakhulu. Uma kuqhathaniswa namanye ama-TCA kanye nesigaba se-SSRI sama-anti-depressants, i-tianeptine powder cishe ayinakho imiphumela emibi. Naphezu kohlelo lwaso lomphumela ophansi, kubalulekile ukungalingani ne-tianeptine ne-monoamine oxidase inhibitors noma ezinye izidakamizwa zokucindezeleka njengoba inhlanganisela ingasongela ukuphila. I-tianeptine akufanele iphinde ixutshwe ne-anesthetics futhi ukusetshenziswa kwayo kufanele kuphele i-24-48 ngaphambi kokungenela okuhlinzekwa okudinga ukuhlinzeka ngezinzwa noma i-hypnotics. Nazi eminye imiphumela emibi ejwayelekile ehambisana ne-tianeptine.

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