I-Raw Tianeptine powder (66981-73-5) ividiyo
I-Raw Tianeptine powder (66981-73-5)
I-Raw Tianeptine powder iyinhlangano ephikisana nokucindezeleka enephrofayli ye-neurochemical novel. I-Raaw Tianeptine powder ayibonakali ihlotshaniswa nokuhlukumezeka kwengqondo, ingqondo, ukulala, imiphumela ye-cardiovascular noma ye-bodyweight futhi inomzimba ophansi wokuhlukunyezwa. I-Raw Tianeptine powder inephrofayli ye-pharmacokinetic ehle kakhulu. Akuhambisani nokuqala kwesimiso se-hepatic, esine-bioavailability ephezulu nokusabalalisa okulinganiselwe, futhi isuswa ngokushesha. Nakuba lokhu kunikeza izinzuzo ze-Raw Tianeptine powder phezu kwama-tricyclic anti-depressant agents ngokusho kwe-dose, izinguquko zokwelashwa kanye nokusebenzisana kwezidakamizwa okungenzeka, ukususwa kwayo ngokushesha kwenza ukunamathela kwamashejuli amaminithi kubaluleke nakakhulu. I-Raw Tianeptine i-powder ihluke kuningi lezinkinga zokulwa nokucindezeleka ngoba akuyona imetabolised uhlelo olusha lwe-cytochrome P450, olubonisa amathuba amancane okusebenzisana kwezidakamizwa; lokhu kunesithakazelo ngokukhethekile iziguli ezigugile.
Imininingwane ye-Raw Tianeptine powder (66981-73-5) Imininingwane
Igama Product | I-Raw Tianeptine powder |
Igama leKhemikhali | I-Raw Tianeptine powder; 66981-73-5; 72797-41-2; I-Raw Tianeptine powder Acid; I-Raw Tianeptine powder |
Brand NAme | I-Yocon |
I-Drug Class | iziphazamiso ezicindezelayo |
CAS Inombolo | 66981-73-5 |
InChIKey | I-JICJBGPOMZQUBB-UHFFFAOYSA-N |
I-molecular Fi-ormula | C21H25ClN2O4S |
I-molecular Weziyisishiyagalombili | I-436.951 g / mol |
IMisa ye-Monoisotopic | I-436.122 g / mol |
Ukuxuba Pi-oint | 148 |
ukubila Point | 609.2 |
I-Half Half-Life | Ayikho idethi etholakalayo |
Color | Mhlophe uphawuda omhlophe |
Sukufaneleka | Ayikho idethi etholakalayo |
Sukuhlushwa Tukushisa | Isiqandisisi |
Aukuphikisana | Kuyisidakamizwa esetshenziselwa ukwelapha iziqephu ezinkulu zokucindezeleka (okuncane, okulinganiselayo, noma okunzima). |
I-Raw Tianeptine powder (66981-73-5) Incazelo
I-Tianeptine powder iyisidakamizwa esetshenziswa kakhulu ekuthuthukiseni izimpawu zengcindezi enkulu yokucindezeleka (MDD). Kuye kwasetshenziselwa ukusiza ukucasula isifo sofuba nesifo se-asthma. Ngokwemvelo, ihlukaniswa ngokuthi i-tricyclic antidepressant (TCA), noma kunjalo, inempahla ehlukile yezokwelapha kunezindlela ezivamile zokulwa nokucindezeleka kwama-tricyclic. I-Tianeptine yatholakale futhi yenziwe i-patented ngumphakathi waseFrance wezokwelapha kwezokwelapha ku-1960s. Amagama omkhiqizo afaka iStablon, Coaxil. ITatinol, Tianeurax, neSalymbra.
I-tianeptine powder ayibonakali ihlotshaniswa nokuhlukumezeka okungaqondakali, ingqondo, ukulala, imiphumela ye-cardiovascular noma bodyweight futhi inomthamo ophansi wokuhlukunyezwa. I-Raw Tianeptine powder inephrofayli ye-pharmacokinetic ehle kakhulu. Akuhambisani nokuqala kwesimiso se-hepatic, esine-bioavailability ephezulu nokusabalalisa okulinganiselwe, futhi isuswa ngokushesha. Nakuba lokhu kunikeza izinzuzo ze-Raw Tianeptine powder phezu kwama-tricyclic anti-depressant agents ngokusho kwe-dose, ukuguqulwa kokwelashwa kanye nokusebenzisana kwezidakamizwa okungenzeka, ukususwa kwayo ngokushesha kwenza ukunamathela kumashejuli amaminithi kubaluleke nakakhulu. I-Raw Tianeptine i-powder ihluke kuningi lezinkinga zokulwa nokucindezeleka ngoba akuyona imetabolised uhlelo olusha lwe-cytochrome P450, olubonisa amathuba amancane okusebenzisana kwezidakamizwa; lokhu kunesithakazelo ngokukhethekile iziguli ezigugile.
Muva nje, i-Tianeptine iyatholakala emazweni aseYurophu, ase-Asia, naseNingizimu Melika. Ivinjelwe e-United Kingdom futhi ayinakekelwa ngokomuthi odokotela base-United States.
I-Tianeptine powder (66981-73-5) Indlela Yokusebenza
Ucwaningo lwamuva lubonisa ukuthi i-tianeptine isebenza njenge-agonist egcwele ku-receptionor ye-opioid (MU). I-receptors yama-opioid njengamanje ihlolisiswa njengenhloso ephumelelayo yezokwelapha ezicindezelayo. Kukholelwa ukuthi imiphumela yomtholampilo ye-tianeptine inesidingo sokuguquguquka kwayo kwala ma-receptors. Ngaphezu kwezinyathelo zawo kwi-receptor ye-opioid, izifundo zangaphambilini zikhokhelwe isenzo salo kumphumela we-serotonin receptor dopamine (D2 / 3) nama-receptors we-glutamate.
I-Tianeptine powder ingumuthi oyingqayizivele we-anti-depressant kanye ne-anxiolytic okhuthaza ukutholwa kwe-serotonin (5-hydroxytryptamine; 5-HT), ne-5-hydroxyindoleacetic acid (5-HIAA) ezicutshini zobuchopho.
Nakuba i-serotonin ye-monoaminergic neurotransmitters (i-5-HT), i-noradrenaline (NA) ne-dopamine (DA) ikhonjiswe ukuthi ihlobene nokuvela kwezinkinga zokucindezeleka, manje sekuqaphele ukuthi ukulahlekelwa kwe-monoamine akwanele ukuchaza indlela yokwenza i-anti-depressant imithi.
Isicelo se-Tianeptine powder (i-66981-73-5)
▪ I-tianeptine ithuthukisa izimpawu zesifo sokucindezeleka esikhulu (MDD)
▪ I-tianeptine isiza isifo samathumbu nesifuba somoya
▪ I-tianeptine ithuthukisa imizwa futhi idambise ukukhathazeka.
▪ I-tianeptine inyusa ukuthi ubuchopho buthatha malini i-serotonin
▪ I-Tianeptine ithuthukisa ukugqugquzela, ukugxila kanye nokuqonda, ukucindezela ukukhathazeka, ukuvuselela amandla nokunciphisa ukukhathala kwengqondo.
Kunconywe i-Tianeptine powder (i-66981-73-5) Isilinganiso
I-tianeptine powder ngokuvamile inqunywa kumthamo we-12.5 mg futhi ithathwa kathathu ngosuku. Ngokungafani namanye ama-TCA kanye nama-serotonin reuptake inhibitors (SSRIs) akhethiwe, imithamo ye-tianeptine ayidingi ukwandiswa kancane futhi i-taper lapho umuthi unqanyuliwe awudingeki.
Imiphumela emibi ye-Tianeptine powder (66981-73-5)
Imiphumela emibi ye-tianeptine powder ikhawulelwe ngokumangazayo. Uma kuqhathaniswa namanye ama-TCA kanye nesigaba se-SSRI se-anti-depressants, i-tianeptine powder cishe ayinayo imiphumela emibi. Naphezu kwephrofayili yayo yomthelela omubi, kubalulekile ukuthi ungaxubi i-tianeptine ne-monoamine oxidase inhibitors noma amanye ama-anti-depressants njengoba inhlanganisela ingasongela impilo. I-Tianeptine akufanele futhi ixutshwe ne-anesthetics futhi ukusetshenziswa kwayo kufanele kuyeke i-24-48 ngaphambi kokungenelela kokuhlinzwa okudinga i-anesthetics noma i-hypnotics. Nayi eminye imiphumela emibi ejwayelekile ehambisana ne-tianeptine.
▲ ukuqunjelwa
▲ Uhudo
▲ Ukuzithoba
▲ Ukuvota
▲ Umlomo omile
▲ Ukukhathala
▲ Insomnia
▲ Izinguquko ekudleni
▲ isiyezi
▲ Ukucindezeleka kokuphefumula
▲ Ukulala
▲ Umbono ophundlekile
▲ Ukunciphisa ukushayela ucansi
▲ bekhanda
▲ Itching