I-Raw Lorcaserin powder (616202-92-7) ividiyo
I-Raw Lorcaserin powder (616202-92-7) Incazelo
I-Lorcaserin powder enomsoco ingokwezigaba zemithi eyaziwa ngokuthi i-serotonin receptor agonists.Isebenza ngokukhulisa imizwa yokugcwala ukuze kudliwe ukudla okuncane.I-Raw Lorcaserin powder isetshenziselwa ukuzivocavoca okuvunyelwe udokotela, ukuguqulwa kokuziphatha, kanye nenhlelo yokunciphisa ikhalori ukukusiza ukuthi ulahlekelwe isisindo. Isetshenziswa abantu abathile ngokweqile, njengalabo abakhuluphele noma abanezinkinga zezokwelapha ezihlobene nesisindo. Ukulahlekelwa isisindo nokuyiyeka kunganciphisa izingozi eziningi zempilo eziza nokukhuluphala, kuhlanganise nesifo senhliziyo, isifo sikashukela, umfutho wegazi ophakeme nokuphila okufutshane.
I-Raw Lorcaserin powder iyi-5-HT2C receptor agonist ekhethiwe, futhi ukuhlolwa kwe-vitro komuthi kukhombise ukukhetha okufanelekile kwe-5-HT2C ngaphezulu kwezinye izinhloso ezihlobene. i-plexus, i-cortex, i-hippocampus, i-cerebellum, i-amygdala, i-thalamus, ne-hypothalamus. Ukusebenza kwama-receptors we-5-HT2C ku-hypothalamus kufanele kusebenze ukukhiqizwa kweproopiomelanocortin (POMC) futhi ngenxa yalokho kukhuthaze ukuncipha kwesisindo. Ucwaningo olwenziwe emitholampilo lukhombisa ukuthi umuthi unganciphisa isisindo sokukhuluphala kanye neziguli ezikhuluphele ngokweqile, ungathuthukisa imingcele yemetabolism ehlobene nokukhuluphala, futhi ubekezelela kahle. Ukusondelana kwe-Raw Lorcaserin powder kwe-5-HT2c 5 izikhathi eziphakeme kune-2-HT100B (ingozi yesifo senhliziyo ye-valvular), inokuphepha okuhle, iyisidakamizwa sokuqala sokulahlekelwa isisindo esivunyelwe yi-FDA ngemuva kuka-5. Ngonyaka we-Raw Lorcaserin powder treatment, isilinganiso sokuncipha kwesisindo sisuka ku-2 kuye kumaphesenti we-1999.
Imininingwane ye-Raw Lorcaserin powder (616202-92-7) Imininingwane
Igama Product | I-Lorcaserin Base powder Base |
Igama leKhemikhali | Raw Lorcaserin powder;(R)-8-Chloro-1-methyl-2,3,4,5-tetrahydro-1H-3-benzazepine |
Brand NAme | Belviq |
I-Drug Class | i-serotonin receptor agonists |
CAS Inombolo | 616202-92-7 |
InChIKey | I-XTTZERNUQAFMOF-QMMMGPOBSA-N |
I-molecular Fi-ormula | C11H14ClN |
I-molecular Weziyisishiyagalombili | 195.69 |
IMisa ye-Monoisotopic | 195.0814772 |
Ukuxuba Pi-oint | Ayikho idatha etholakalayo |
Fukuvuselela kabusha Pi-oint | Ayikho idatha etholakalayo |
I-Half Half-Life | Ukuphila kwengxenye ye-plasma cishe amahora angu-11. |
Color | powder emhlophe |
solubility | Ukunwebeka kwamanzi kunkulu kune-400 mg / mL. |
Storage Tukushisa | -20 ℃ Freezer |
Aukuphikisana | Ukuze ukwelashwa ngokweqile, njengokuhambisana nokudla okuncishisiwe-khalori nokusebenza komzimba okwandisiwe. |