I-MT2 (i-Melanotan-II) i powder (i-121062-08-6) ividiyo
I-MT2 (i-Melanotan-II) i powder (121062-08-6) Incazelo
I-Melanotan II (MT-2) iyi-peptide eyenziwe, i-analogue ye-hormone yemvelo ethuthukisa i-melanocortin tan (ukukhiqizwa kwe-melanin ngokusebenzisa i-melanocyte, enquma futhi yenze sikwazi ukusha), ngaleyo ndlela inciphise ingozi yokulimala kwelanga nokunye imiphumela elimazayo yemisebe yelanga ne-solarium.
Le peptide MT-2 yenzelwe ukukhuthaza kakhulu ukusabela komzimba ekuvezweni kwe-UV ray, ngoba ukukhiqizwa kwe-melanin kukhululeke kakhulu ukutholakala kwelanga kuyadingeka ukuthola umphumela omkhulu wokushuka. Lesi yisixazululo esihle kulabo abanesikhumba esifanelekile ukuba bashukwe ngaphandle kokuchitha amasonto elangeni futhi badlule kwinqubo yokusha nokuphulukisa.
Abasebenzisi beMT2 babona ukushuka okusheshayo nokuphulukiswa okusheshayo kwamaseli esikhumba elimele ilanga. Ngenxa yalokhu, i-melanotan II ilungele ikakhulukazi labo abanesikhumba esiphaphathekile (uhlobo lwesikhumba 1 & 2) futhi bathambekele ekushisweni yilanga.
Ngokuqondene nomthamo we-Melanotan II, inqubo yokwamukela ejwayelekile isho ukuthatha umthamo owodwa womjovo we-Melanotan II enanini le-1 mg (ukubalwa ngqo kwekhilogremu ngalinye akudingeki, njengoba imithamo ihlukahluka kakhulu), qala nge-250mkg ngosuku nangezinsuku ze-4 engeza enye i-250mkg kancane. Ngosuku lwesine khuphula umthamo ufike ku-1mg futhi unamathele kuleli zinga kuze kube yilapho kutholakala isifiso esifunekayo. Imininingwane eminingi mayelana nokuthenga uMelanotan II (MT-2) online, sicela ungangabazi ukukhuluma nathi umphakeli we-peptide.
I-MT2 (i-Melanotan-II) i powder (121062-08-6) Siziqu
Igama Product | I-MT2 (i-Melanotan-II) enamandla |
Igama leKhemikhali | I-Melanotan II; I-MelanotanII;
(3S,6S,9R,12S,15S,23S)-12-((1H-imidazol-5-yl)methyl)-3-((1H-indol-3-yl)methyl)-15-((S)-2-acetamidohexanamido)-9-benzyl-6-(3-guanidinopropyl)-2,5,8,11,14,17-hexaoxo-1,4,7,10,13,18-hexaazacyclotricosane-23-carboxamide |
ukulandelana | I-Ac-Nle-cyclo (i-Asp-His-DPhe-Arg-Trp-Lys) -NH2 |
Brand NAme | N / A |
I-Drug Class | Peptide |
CAS Inombolo | 121062-08-6 |
InChIKey | I-JDKLPDJLXHXHNV-MFVUMRCOSA-N |
I-molecular Fi-ormula | C50H69N15O9 |
I-molecular Weziyisishiyagalombili | I-1024.198 g / mol |
IMisa ye-Monoisotopic | I-1023.54 g / mol |
Ukuxuba Pi-oint | > 181 ° C (subl.) |
Fukuvuselela kabusha Pi-oint | ≥17.0 |
I-Half Half-Life | 33 ihora |
Color | White |
Sukufaneleka | I-Soluble ku-DMSO |
Sukuhlushwa Tukushisa | -20 ° C |
Aukuphikisana | I-Melanotan II i-acetate usawoti isetshenziselwe ukutadisha imiphumela yayo yokuvimbela ekusetshenzisweni kokudla nokusetshenziswa kwamandla kwamagundane.
I-Melanotan II i-Acetic Acid Salt, iyimakhemikhali eyenziwe nge-lab efana ne-hormone etholakala kubantu. I-Melanotan II iboniswe ukuthi ine-melanogenesis (ukuthungula) nemiphumela ye-aphrodisiac kubantu. |