I-Nooglutyl powder enomsoco (112193-35-8) ividiyo
I-Nooglutyl powder ephezulu (112193-35-8) Incazelo
I-Nooglutyl powder enomsoco i-agent e-nootropic eyacwaningwa ku-Research Institute of Pharmacology, i-Russian Academy of Medical Sciences njengendlela yokwelashwa okungenzeka ibe yinkinga ye-amnesia. Ezilwaneni zezilwane, kunezinhlobonhlobo zemiphumela yesistimu ephakathi.
I-Nooglutyl powder emnyama (112193-35-8) Siziqu
Igama Product | I-Nooglutyl powder |
Igama leKhemikhali | I-Nooglutil; I-ONK-10; UNII-09UM5JOS3W; I-BRN 4200454; 09UM5JOS3W; I-N-5- (Hydroxynicotinoyl) -l-glutamic acid Okuningi… |
Brand NAme | I-Nooglutil |
I-Drug Class | Izidakamizwa zeNootropic |
CAS Inombolo | 112193-35-8 |
InChIKey | I-XFZGYOJFPGPYCS-QMMMGPOBSA-N |
I-molecular Fi-ormula | C11H12N2O6 |
I-molecular Weziyisishiyagalombili | 268.225 g |
IMisa ye-Monoisotopic | 268.23 g / mol |
ukubila Point | I-704.7 ± 60.0 ° C ku-760 mmHg |
Fukuvuselela kabusha Pi-oint | N / A |
I-Half Half-Life | Imizuzu ye-30 kumahora angu-3 |
Color | powder emhlophe |
Sukufaneleka | kancane incibilika emanzini nase-ethanol. |
Sukuhlushwa Tukushisa | Gcina ekamelweni lokushisa, emgodini ovalwe, gwema ukushisa okuqinile nokukhanya. |
Aukuphikisana | I-Nooglutyl powder ewusizo i-nootropic entsha esinikeza ukugcinwa kwememori evelele nokukhumbula izinzuzo. |
Raw I-Nooglutyl powder (112193-35-8) Incazelo
I-Nooglutyl powder iyinkampani ye-nootropic efundiswa ku-Research Institute of Pharmacology, i-Russian Academy of Medical Sciences njengendlela yokwelapha i-amnesia.Izibonelo zezilwane, kunezimo ezihlukahlukene zesistimu yezinzwa zomphakathi.
I-Nooglutyl, eyakhiwe yi-L-glutamic ne-oxynicotinic acid, enemiphumela ye-glutamatergic iyisidakamizwa esisebenzayo kakhulu ekuphatheni ukuphazanyiswa kwememori nokufunda, ukuvikela umonakalo we-ischemic neuronal nokulimala komqondo. Tere
I-Nooglutyl powder (112193-35-8) Inqubo yesenzo?
Ukuhlolwa kwamagundane kubonisa ukuthi i-nooglutyl ibonisa izakhiwo ezivikela izidakamizwa kanye nomsebenzi wayo wokulwa ne-antimotion ayifaki ngaphansi kwezivikeli zangasese ezingezansi, njenge-scopolamine ne-diprazine. Ukuhlolwa kwe-electrophysiological kwamakati kubonisa ukuthi i-nooglutyl ishintshela umsebenzi owenziwe ngokuzenzakalelayo ku-80% ye-neurons yama-cortical (indawo engezansi ye-somatosensory I ne-5 ye-parietal association cortex) futhi iyanciphisa kakhulu imiphumela ebangelwa ukugula okuhambayo: ukusebenza komsebenzi owodwa we-unit of zone somatosensory I nokuvimbela izimpendulo ze-neuron ekugqugquzelweni kwe-somatic. Le ndawo yokulungiswa ikholelwa ukuthi yakha isisekelo somphumela wayo wokulwa nezidakamizwa.
I-Nooglutyl iye yaboniswa ngokukhetha i-AMPA receptors, ejwayelekile ye-ampakine stimulant, ngezici ze-neuroprotective ze-racetam. Kuye kwaboniswa ukuthi kunomthelela onamandla kuma-receptors we-glutamate kunoNoopept.
Izinzuzo of I-Nooglutyl powder (112193-35-8)
Kungcono kwi-Memory Creation nokugcinwa
I-nooglutyl powder inqunyelwe ukuba ibe nezakhiwo ze-nootropic eziphumelelayo nezamandla. I-Nooglutyl yaqaphela ukuthi ibe nomthelela omuhle ekudalweni kwememori nokugcinwa, futhi nayo yakwazi ukuthuthukisa iningi lezinqubo zokucatshangelwa zezilwane zelabhu. Ucwaningo lubuye lwaphakamisa ukuthi lwalunezimpawu zokulwa namagciwane.
Kunconywe I-Nooglutyl powder (112193-35-8) Isilinganiso
Ayikho incomo yokuncoma kumuntu okwamanje, kodwa i-Nooglutyl powder esilinganisweni se-20 mg / kg ikhiqiza umphumela omuhle ekuphatheni nasekukhunjweni kwamagundane omdala we-SAMP9 we-10.
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